Manufacturer: Focus Biomolecules
Second generation oral hypoglycemic agent. Acts via ATP-dependent K+ channel (Kir6, KATP) block1. Inhibits Kir6 currents in the pancreas, causing an increase in intracellular Ca2+ and insulin secretion. Also inhibits recombinant CFTR Cl- channels with an IC50 of 20 μM2. Cell permeable.
CAS Number: 10238-21-8
Manufacturer Part Number/SKU: 10-1325-5g-EA
Tags: Focus Biomolecules