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GSK2879552, LSD1 inhibitor, 5mg, CAS# 1401966-69-5

$80.00
4-[[4-[[[(1R,2S)-2-Phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]benzoic acid dihydrochloride Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )

Manufacturer: Focus Biomolecules

SKU
10-4020-5mg-EA
GSK2879552, LSD1 inhibitor, 5mg, CAS# 1401966-69-5 is available to buy in increments of 1

Product Details

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GSK289552 is potent, selective, and irreversible inhibitor of Lysine Demethylase 1 (LSD1) via covalent modification of the LSD1 cofactor FAD (Ki = 1.7 µM). It is selective for LSD1 over the closely related LSD2, MAO-A, MAO-B, and the FAD dependent enzymes D-amino acid oxidase and glutathione reductase. Tested against a panel of 165 cancer cell lines, GSK2879552 inhibited the proliferation of 9 small cell lung carcinoma lines and 20 AML cell lines.

CAS Number: 1401966-69-5

Manufacturer Part Number/SKU: 10-4020-5mg-EA

Tags: Focus Biomolecules