Manufacturer: Focus Biomolecules
Potent and selective PARP-inhibitor with Ki values of 5.2 nM and 2.9 nM for PARP-1 and PARP-2, respectively.1 Restores sensitivity to DNA alkylator/methylator temozolomide in glioma cells and xenografts2, and enhances radiotherapy sensitivity in endometrial carcinoma cells3. Also improves sensitivity to DNA replication inhibitor cisplatin in human oral carcinoma cells.4
CAS Number: 912445-05-7
Manufacturer Part Number/SKU: 10-2419-25mg-EA
Tags: Focus Biomolecules