UNC6934, NSD2 inhibitor, 25mg, CAS# 2561494-77-5
$210.00
N-Cyclopropyl-3-oxo-N-(4-pyrimidin-4-ylcarbamoyl)benzyl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-7-carboxamide Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )
Manufacturer: Focus Biomolecules
SKU
10-4119-25mg-EA
UNC6934, NSD2 inhibitor, 25mg, CAS# 2561494-77-5 is available to buy in increments of 1
Product Details
Download Details and SpecificationsPotent (IC50 = 104 nM) and selective inhibitor of protein lysine methyltransferase nuclear receptor-binding SET domain-containing 2 (NSD2). It potently binds to the PWWP1 domain antagonizing interaction with nucleosomal H3K36me2. UNC6934 is selective against 14 other human PWWP domains and 33 methyltransferases. Active in a nanoBRET PPI assay in U2OS cells (IC50 = 1.23 µM).
CAS Number: 2561494-77-5
Manufacturer Part Number/SKU: 10-4119-25mg-EA
Tags: Focus Biomolecules