Manufacturer: Focus Biomolecules
Potent and selective antagonist of the TRPV1 receptor (IC50's for receptor induction method: Capsaicin = 3 nM; Acid (pH5.3) = pIC50 7.1, and Heat = 6 nM) with activity in human, rat, and guinea pig receptors.1,2 SB-705498s activity is voltage dependent and shows >100 fold selectivity over the closely related TRPM8 receptor.2
CAS Number: 501951-42-4
Manufacturer Part Number/SKU: 10-3985-25mg-EA
Tags: Focus Biomolecules