S1RA, Sigma-1 antagonist, 5mg, CAS# 1265917-14-3
$85.00
4-{2-[5-Methyl-1-(napthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine hydrochloride Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )
Manufacturer: Focus Biomolecules
SKU
10-4201-5mg-EA
S1RA, Sigma-1 antagonist, 5mg, CAS# 1265917-14-3 is available to buy in increments of 1
Product Details
Download Details and SpecificationsS1RA (E-52862) is a potent and selective s1 antagonist with weak binding at s2 (IC50's: s1 = 17nM, s2 = 9300nM).1,2 S1RA abolished mechanical and thermal hyperalgesia in mice with carrageenan-induced acute inflammation by enhancing the action of endogenous opioid peptides of immune origin in a s1 dependent manner.3 BD1063 potentiated µ-opioid antinociception in mice in a s-dependent manner.4 S1RA displayed neuroprotective effects in a mouse model of ischemic stroke.5
CAS Number: 1265917-14-3
Manufacturer Part Number/SKU: 10-4201-5mg-EA
Tags: Focus Biomolecules