Manufacturer: Focus Biomolecules
MU1700 is a potent (IC50's = 13 nM ALK1; 6 nM ALK2) and highly selective (selective against 369 kinases with only ALK6 (41 nM) being inhibited) ALK1/2 inhibitor. Much higher kinome selectivity than the typically used ALK 1/2 inhibitor LDN-193189. MU1700 exhibits favorable pharmacokinetic and bioavailability profiles for in vivo use. It showed excellent CNS penetration with brain concentrations exceeding that in plasma.
CAS Number: 1360905-04-9
Manufacturer Part Number/SKU: 10-4746-5mg-EA
Tags: Focus Biomolecules