GSK-1016790A, TRPV4 channel blocker, 5mg, CAS# 942206-85-1
$68.00
(N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide Purity: 98% by TLC Purity: NMR (Conforms) Store -20°C Ship RT (1 per EA )
Manufacturer: Focus Biomolecules
SKU
10-1198-5mg-EA
GSK-1016790A, TRPV4 channel blocker, 5mg, CAS# 942206-85-1 is available to buy in increments of 1
Product Details
Download Details and SpecificationsA novel and potent TRPV4 channel agonist. GSK1016790A induced Ca2+ influx in mouse and human TRPV4 expressing HEK cells (EC50 values of 18 and 2.1 nM, respectively), and evoked a dose-dependent activation of TRPV4 whole-cell currents at concentrations above 1 nM. It is 300-fold more potent than 4α-PDD and is a valuable tool for investigating the role of TRPV4 in physiological processes.
CAS Number: 942206-85-1
Manufacturer Part Number/SKU: 10-1198-5mg-EA
Tags: Focus Biomolecules