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Fruquintinib, VEGFR kinase inhibitor, 5mg, CAS# 1194506-26-7

$60.00
6-(6,7-Dimethoxyquinazolin-4-yl)oxy-N,2-dimethyl-1-benzofuran-3-carboxamide Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )

Manufacturer: Focus Biomolecules

SKU
10-4784-5mg-EA
Fruquintinib, VEGFR kinase inhibitor, 5mg, CAS# 1194506-26-7 is available to buy in increments of 1

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Fruquintinib is a potent and highly selective inhibitor of VEGFR kinase (IC50's: VEGFR1= 33 nM, VEGFR2 = 35 nM, VEGFR3 = 0.5 nM).1 It potently inhibited VEGF/VEGFR signaling and cell proliferation in HUVECs and HLECs and prevented angiogenesis in vitro. Fruquintinib is currently is several clinical trials against metastatic colorectal cancer2 and nonsquamous non-small-cell lung cancer3.

CAS Number: 1194506-26-7

Manufacturer Part Number/SKU: 10-4784-5mg-EA

Tags: Focus Biomolecules