EED-226, PRC2 methyltransferase inhibitor, 25mg, CAS# 2083627-02-3

EED-226, PRC2 methyltransferase inhibitor, 25mg, CAS# 2083627-02-3

PTC-209, BMI-1 inhibitor, 5mg, CAS# 315704-66-6

PTC-209, BMI-1 inhibitor, 5mg, CAS# 315704-66-6

EED-226, PRC2 methyltransferase inhibitor, 5mg, CAS# 2083627-02-3

$65.00
N-(Furan-2-ylmethyl)-8-(4-methylsulfonylphenyl)-[1,2,4]triazolol[4,3-c)pyrimidine-5-amine Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )

Manufacturer: Focus Biomolecules

SKU
10-4021-5mg-EA
EED-226, PRC2 methyltransferase inhibitor, 5mg, CAS# 2083627-02-3 is available to buy in increments of 1

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EED-226 is a potent (IC50 = 23.4 nM) and selective allosteric inhibitor of the EED subunit of the methyltransferase polycomb repressive complex 2 (PRC2).1,2 It caused drastic proliferation inhibition in lymphoma cells with EZH2 mutations and caused shrinkage and slower tumor growth in mice using a subcutaneous xenograft model of Karpas422.

CAS Number: 2083627-02-3

Manufacturer Part Number/SKU: 10-4021-5mg-EA

Tags: Focus Biomolecules