CPI203, BET bromodomain inhibitor, 25mg, CAS# 1446144-04-2
$350.00
(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6h-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamide Purity: 98% by HPLC NMR (Conforms) Store -20°C Ship RT (1 per EA )
Manufacturer: Focus Biomolecules
SKU
10-4048-25mg-EA
CPI203, BET bromodomain inhibitor, 25mg, CAS# 1446144-04-2 is available to buy in increments of 1
Product Details
Download Details and SpecificationsCPI203, a JQ1 analog, is a potent and selective inhibitor of the BET bromodomain BRD4 (IC50 = 26 nM).1 It helps promote the maintenance of hematopoietic stem cells via repression of Myc expression.2 CPI203 reversibly suppressed intestinal stem cell differentiation in a mouse model.3 It enhanced the expansion of human cord blood hematopoietic stem cells without losing cell viability.4 CPI203 displays synergistic antitumor activity with various agents including lenalidomide5, bortezomib6, and PARP inhibitors7.
CAS Number: 1446144-04-2
Manufacturer Part Number/SKU: 10-4048-25mg-EA
Tags: Focus Biomolecules