BI-6015, HNF4α inhibitor, 5mg, CAS# 93987-29-2
$50.00
2-Methyl-1-[(2-methyl-5-nitrophenyl)sulfonyl]-1H-benzimidazole Purity: 98% by TLC Purity: NMR (Conforms) Store -20°C Ship RT (1 per EA )
Manufacturer: Focus Biomolecules
SKU
10-1402-5mg-EA
BI-6015, HNF4α inhibitor, 5mg, CAS# 93987-29-2 is available to buy in increments of 1
Product Details
Download Details and SpecificationsHepatocyte nuclear factor 4α (HNF4α) antagonist. HNF4α is a central regulator of gene expression in cell types that play a central role in metabolic homeostasis. 1 BI-6015 binds to HNF4α with high affinity and modulates the expression of known target genes. It was shown to be selectively cytotoxic to cancer cell lines in vitro and in vivo however in vivo potency was limited by suboptimal pharmacokinetics. 2 Represents the first small molecule tool for pharmacologic modulation of HNF4α activity. 2 Cell permeable.
CAS Number: 93987-29-2
Manufacturer Part Number/SKU: 10-1402-5mg-EA
Tags: Focus Biomolecules