Manufacturer: Focus Biomolecules
Potent and selective inhibitor of PI 3-kinase g (PI 3-K g ), IC50 = 8 nM displaying 30-fold selectivity over PI 3-Kd and PI 3-Kb and 7.5-fold selectivity over PI 3-Ka1. Suppresses joint inflammation in two distinct mouse models1. Ameliorates surgical brain injury2, colitis3, intimal hyperplasia-induced inflammatory processes4 and renal injury/fibrosis5 in rodent models. Orally active.
CAS Number: 648450-29-7
Manufacturer Part Number/SKU: 10-2575-25mg-EA
Tags: Focus Biomolecules