Manufacturer: Focus Biomolecules
Alpelisib is a potent and selective (IC50s = 7.4 nM PI3Kα; 2.2 µM PI3Kß; 1.2 µM PI3KIδ; 50-fold selectivity against 442 tested kinases) PI3Kα inhibitor.1 Approved for use in the treatment of HR(+), HER2(-), PIK3CA-mutated breast cancer. Alpelisib has been used in combination with various chemotherapeutics to treat ovarian2, colorectal3, kidney4, bladder5, and head and neck6 cancers.
CAS Number: 1217486-61-7
Manufacturer Part Number/SKU: 10-4167-5mg-EA
Tags: Focus Biomolecules